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Angiotensin Converting Enzyme Inhibitors

Action

Hydrolyzed to active form which inhibit conversion of angiotensin I to angiotensin II (potent vasoconstrictor) Meabolism By liver

Elimination Mainly via urine; Indication HT LV dysfunction Congestive heart failure Renal impairment

Side Effects Hypotention Dry cough Risk of hyperkalemia Rash, angioedema Contra-indication Bilateral renal artery stenosis Hypersensitivity. Pregnancy.

e.g.
Captopril Enalapril Ramipril

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