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Rumus kimia3
Kodein
Efek analgesiknya
lebih rendah
dibanding morfin.
Tidak menimbulkan
depresi
pernafasan.
Morfin
Farmakokinetik 2
Dosis 1
Onset of action:
Oral: 0.5-1 hour;
I.M.: 10-30 minutes
Peak effect: Oral:
1-1.5 hours; I.M.:
0.5-1 hour
Duration: 4-6 hours
Absorption: Oral:
Adequate
Distribution:
Crosses placenta;
enters breast milk
Protein binding: 7%
Metabolism:
Hepatic to
morphine (active)
Half-life
elimination: 2.5-3.5
hours
Excretion: Urine
(3% to 16% as
unchanged drug,
norcodeine, and
free and
conjugated
morphine)
DEWASA :
IM/perlahan IV/SC
15-60 mg tiap 4-6
jam (maksimum
360 mg/hari). (A to
Z)
IV 2,5-15 mg / 70
kg dalam 4 sampai
5 ml WFI lebih dari
5 menit prn. IV (MI
nyeri) 8 sampai 15
(+)/(-)4
Harga 5