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Indikasi Tambahan
bradycardy, cardiogenic shock,
Potensi Efek Samping hypotension,raynaud's syndrome,
dizziness, death
hypersensitivity, uncompensated
congestive heart failure.
Kontra indikasi
Cardiogenic shock, bradycardy,
COPD.
Peringatan
Dosis
Frekuensi pemberian 2 - 3 / day
Harga
Arbutamine / selected
Potensi interaksi obat
antiarrhytmics (severe interaction)
Hypertrophic obstructive
Kondisi yang berpotensi meningkatkan risiko efek samping
cardiomyopathy; dysrhytmias
TUTOR 17 / E1
7-9 hari 21 hr
highly lipophilic, hampir semua poorly absorbed from the GI
100%
diabsorpsi setelah administrasi oral tract and low bioavailability.
hipersensitif ke acetylcholine
hipersensitivitas, ventricular chloride, acute iritis, acute
hypersensitivity, renal failure
fibrilation inflammatory disease di anterior
chamber
1. Aminoglutethimide ( Metabolism
of digitoxin accelerated (reduced Frusemide or Furosemide
Acebutolol, Ambenonium, Bisoprolol, dll. (The risk or severi
effect)) 2. Calcium (can precipitate (menguntungkan/merugikan)
arrhythmias)
Atropine berkompetisi
dengan ACh dan
muscarinic agonist lainnya nonselective beta adrenergic
pada muscarinic receptor. blocker(class II antiarhytmic,
Saat atropine berikatan memblok reseptor alfa- competitively block response
menstimulasi alpha dan
dengan reseptor adrenergik, di samping beta 1 and beta 2 adrenergic
beta 1 adrenergic
muscarinic, atropine itu juga menstimulasi stimulation which result in
receptor
mencegah pelepasan reseptor β-adrenergic decrease heart rate,
inositol triphosphate (IP3) myocardial contractility and
dan inhibisi adenylyl myocardial oxygen demand.
cyclase yang disebabkan
oleh muscarinic agonist.
- menurunkan kontraksi
anaphylactic shock,
sepsis,cardiac arrest,
Parkinson’s disease, motion
resistant ventricular pasien penderita hypertension, angina pectoris,
sickness, ophthalmologic
fibrillation,bronchospas hipertensi yang terjadi phreocomochytoma, essential
disorder, COPD, asthma,
m, severe asthma, dalam rangkaian tremor, supraventricular
minor inflammatory
unresponsive asystole, persitiwa yang arhytmia, ventricular
bladder disorder,
unresponsive disebabkan oleh tachycardy, prevention of MI,
cholinergic poisoning,
bradychardia, pheochromacytoma migrain.
bradycardia
laryngotracheobronchiti
s
hypertensive crisis,
pheochromocytomas,
in adjunctive therapy of necrosis caused by
Hyperhidrosis
anesthesia administration site
extravasation,
norepinephrine
sweating, nausea,
vomit, headache,
chestpain,
hypertension,
Mydriasis, cycloplegia, dry hyperglycemia, acute and prolonged
mouth, tachycardia, hot and hypokalemia, cardiac hypotensive episodes, bradycardy, cardiogenic shock,
flushed skin, agitation, arrythmias, weakness, fast heart rate, cardiac hypotension,raynaud's
delirium, urinary retention, dizziness, anxiety, arrhythmias, weakness, syndrome, dizziness
constipation dyspnea, restlessness, dizziness
palpitation,
tachychardia,tremors,
cold extrimities, susah
buang air kecil
hypertension,
hyperthyroid, Myocardial infarction,
tacharrythmias, history of myocardial
glaucoma, history of ventricular fibrillation, infarction, coronary hypersensitivity,
prostatic hyperplasia, acid- ischemic heart disease, insufficiency, angina or uncompensated congestive
peptic disease, urinary tract angle closure other evidence suggestive heart failure. Cardiogenic
obstruction, GI obstruction galucoma, DM, of coronary artery shock, bradycardy, COPD.
idiopathic hyperthropic disease; hypersensitivity
subaortic stenosis, to Phentolamine
pheochromocytoma
Phentolamine dapat
hati hati pemberian
menyebabkan hipotensi
epinephrine pada orang
akut maupun
tua dan anak anak,
reflux esophagitis, elderly, berkepanjangan,
penyesuaian dosis pada
infants, children takikardia, aritmia,
orang orang yang
angina, infark
mempunyai penyakit
myokardium, dan spasma
ginjal dan hati
serebrovaskular
Phentolamine dapat
menyebabkan hipotensi
akut maupun
berkepanjangan,
IV/IM IV, oral
takikardia, aritmia,
angina, infark
myokardium, dan spasma
serebrovaskular
- tidak tersedia
Phentolamine 84 USD (5
Rp41704
mg vial)
AU TGA pregnancy
category: A US FDA
pregnancy category: C
kategori C Comments: -Use with C C
caution during labor and
delivery; avoid use during
second stage of labor.
aman dengan dosis
yang disesuaikan
tidak direkomendasikan tidak tersedia Enter breast milk
dengan umur dan juga
berat
Diabetes
Glucoma,Reflux Hypotension,Obstructive Acidosis,Asthma,Heart
mellitus,Hypertension,Hy
oesophagitis,Prostatic cardiomyopathy,Cardiovascula failure,Cardiogenic
perthyroidism,Ischaemic
hypertrophy,Unstable cardiac r disease,Cerebrovascular shock,Bronchospasm,Haemorrhage,H
heart disease,Angle- disease,Aortic stenosis. eart block.
rhythm.
closure glaucoma.
Verapamil Isosorbit dinitrate
menurunkan kontraksi
Norverapamil adalah
metabolit verapamil yang
masih mempunyai aktivitas hepatic
farmakodinamik yang
lemah.
dengan makan
Amiodarone (HCl)
(enhance the bradycardic
Quinine (enhance the hypotensive
effect), Amobarbital
effect),
(reduces hypotensive
Carbamazepine, Cimetidine (HCl),
effects ), Betaxolol (HCl)
Clarithromycin (decrease the
(Severe hypotension when
metabolism of Isosorbide(Dinitrate))
and heart failure when beta
blockers)
Hypovolaemia,Myocardial
Heart infarction,Cardiac temponade,Raised
failure,Bradycardia,Platelet intracranial pressure,Low cardiac
dysfunction. output,Obstructive hypertrophic
cardiomyopathy.