Escolar Documentos
Profissional Documentos
Cultura Documentos
2 Sensitizers
2.1 Biguanides
2.2 Thiazolidinediones
2.3 Lyn kinase activators
3 Secretagogues
3.1 Sulfonylureas
First-generation agents
tolbutamide
acetohexamide
tolazamide
chlorpropamide
Second-generation agents
glipizide
glyburide or glibenclamide
glimepiride
gliclazide
glyclopyramide
gliquidone
3.2 Non-sulfonylurea secretagogues
Meglitinides
repaglinide
nateglinide
4 Alpha-glucosidase inhibitors
miglitol
acarbose
voglibose
5 Peptide analogs
molecules that fulfill criteria for being an incretin are
glucagon-like peptide-1 (GLP-1) and gastric inhibitory peptide
(glucose-dependent insulinotropic peptide, GIP). Both GLP-1 and GIP
are rapidly inactivated by the enzyme dipeptidyl peptidase-4 (DPP-4).
5.1 Injectable incretin mimetics
Exenatide
Liraglutide
Taspoglutide
Lixisenatide
Semaglutide
Dipeptidyl peptidase-4 (DPP-4) inhibitors
vildagliptin (Galvus)
sitagliptin (Januvia)
saxagliptin (Onglyza)
linagliptin (Tradjenta)
alogliptin
septagliptin
Teneligliptin
Gemigliptin: Zemiglo
5.2 Injectable amylin analogues
pramlintide
6 Glycosurics
SGLT-2 inhibitors
Dapagliflozin
Canagliflozin
Empagliflozin
7 Comparison
8 Generic