Escolar Documentos
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Receptor type
Dopamine (D2)
Serotonin 1A (5-HT1A)
Serotonin 2A (5-HT2A)
Serotonin 2C (5-HT2C)
Class & MOA
SSRIs: inhibit
reuptake of serotonin
as well as slight
effects on histamineR, 1-R, and
muscarinic-R
SNRIs: inhibits
reuptake of both
serotonin and
norepinephrine
Atypical
Antidepressants
Brand
Prozac
Citalopram
Celexa
Escitalopram
Lexapro
Fluvoxamine
Luvox
Sertraline
Zoloft
Paroxetine
Paxil
Venlafaxine (ER
avail)
Effexor
Duloxetine
Cymbalta
Desvenlafaxine
Bupropion
Pristiq
Wellbutrin
Mirtazapine
Remeron
Nefazodone
Trazodone
Serzone
Oleptro
Generic Agent
Brand
Receptor type
Serotonin 3 (5-HT3)
Alpha-1 adrenergic (-1)
Histamine (H1)
Muscarinic (m1)
Info
Info
Tricyclic
Antidepressants:
inhibits reuptake of
both serotonin and
norepinephrine
MAOIs: block
destruction of
monoamines
centrally and
peripherally
Mood Stabilizers
Amitriptyline
Elavil
Clomipramine
Desipramine
Doxepin
Imipramine
Nortriptyline
Phenelzine
Anafranil
Norpramin
Silenor
Tofranil
Pamelor
Nardil
Tranylcypromine
Parnate
-Irreversible
Selegiline
Emsam
(transdermal)
-Reversible
Carbamazepine
Tegretol
Valproate
Depakene
Depakote
Lamotrigine
Lamictal
Lithium
Eskalith
Lithobid
Gabapentin
Neurontin
Generic Agent
Brand
-Least sedating
-Irreversible
Info
Benzodiazepines:
GABA-R agonists
CNS inhibition
Other Anxiolytics
Typical
Antipsychotics:
nonselective DA-R
antagonists
Atypical
Antipsychotics:
block postsynaptic
DA-R, block
serotonin-R, variable
effect on histaminic
and cholinergic-R
Chlordiazepoxide
Librium
Clorazepate
Diazepam
Flurazepam
Alprazolam
Tranxene
Valium
Dalmane
Xanax
Clonazepam
Klonopin
Lorazepam
Temazepam
Oxazepam
Triazolam
Buspirone
Ativan
Restoril
Serax
Halcion
BuSpar
Haloperidol (inj
avail)
Fluphenazine
Perphenazine
Thioridazine
Haldol
Chlorpromazine
Aripiprazole
Asenapine (SL
tablet avail)
Olanzapine (inj
avail)
Thorazine
Abilify
Saphris
Prolixin
Trilafon
Mellaril
Ziprasidone
Zyprexa
Zyprexa
Relprevv (inj)
Seroquel
Risperdal
Consta (inj)
Geodon
Clozapine
Clozaril
Iloperidone
Fanapt
Lurasidone
Paliperidone (inj
avail)
Latuda
Invega
Invega
Sustenna (inj)
Quetiapine
Risperidone
-Long-acting
-Used often during EtOH withdrawal
-Long-acting
-Long-acting
-Long-acting
-Intermediate acting
-Approved for panic disorder
-Intermediate acting
-Approved for panic disorder
-Intermediate acting
-Intermediate acting
-Short acting
-Short acting
-5-HT partial agonist
-Gradual onset in 2 weeks
-Does not potentiate effects of alcohol = useful in alcohols
-Low addiction potential = good for pts who were addicted to benzos or other drugs
-AEs: sexual, dizziness, nausea, HA
-Drug interactions
-Good for acute agitation as onset is 30 min
Dystonias
-Benztropine
-Biperiden
-Diphenhydramine
-Trihexyphenidyl
Akathisias = restlessness
-Propranolol
-Benzos
Parkinsonianism
-Amantadine
-Levodopa
Extrapyramidal Symptoms
-Parkinsonian syndrome, acute dystonias, akathisia
-Benztropine
-Benadryl